Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 3' and Ligand = 'BDBM50394155'
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50394155(CHEMBL2158814)
Affinity DataKi:  6.31nMAssay Description:Binding affinity to human CCR3 receptor expressed in CHOK1 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50394155(CHEMBL2158814)
Affinity DataKi:  6.31nMAssay Description:Binding affinity to human CCR3 expressed in CHOK1 cells by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50394155(CHEMBL2158814)
Affinity DataIC50:  8.10nMAssay Description:Antagonist activity at CCR3 assessed as inhibition of eotaxin bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50394155(CHEMBL2158814)
Affinity DataKd:  100nMAssay Description:Antagonist activity at CCR3 receptor in human poylmorphonuclear leukocytes assessed as inhibition of eotaxin-induced CD11b expression after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed