Found 4 Enz. Inhib. hit(s) with Target = 'Calcium/calmodulin-dependent protein kinase type II subunit alpha' and Ligand = 'BDBM50163745' TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of autophosphorylated alphaCaMK2 using GST-NR2A as substrate incubated for 1 min prior to substrate addition measured after 1 min in prese...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of alphaCaMK2 using GST-NR2A as substrate incubated for 1 min prior to substrate addition measured after 1 minMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of alphaCaMK2 autophosphorylation at Thr286 using [gamma32P]ATP incubated for 30 secs prior to ATP addition measured after 30 secsMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit alpha(Homo sapiens (Human))
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Rajiv Gandhi Centre For Biotechnology
Curated by ChEMBL
Affinity DataIC50: 2.44E+4nMAssay Description:Inhibition of autophosphorylated alphaCaMK2 using GST-NR2A as substrate incubated for 1 min prior to substrate addition measured after 1 minMore data for this Ligand-Target Pair
