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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50399525'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399525(CHEMBL2180226 | US9187480, tert-butyl 4-{[8-(2-chl...)
Affinity DataKi:  23.9nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399525(CHEMBL2180226 | US9187480, tert-butyl 4-{[8-(2-chl...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed