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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50232933'
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232933(CHEMBL4094388)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation and luminescence co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL
LigandPNGBDBM50232933(CHEMBL4094388)
Affinity DataIC50:  35nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 EBNA cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed