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Found 4 Enz. Inhib. hit(s) with Target = 'Cathepsin K' and Ligand = 'BDBM50148291'
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148291(((S)-1-Formyl-pentyl)-carbamic acid (S)-2-cyclohex...)
Affinity DataIC50:  2.70nMAssay Description:Inhibitory concentration against recombinant human cathepsin K determined in a fluorescence assay using 10 microM Cbz-Phe-Arg-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148291(((S)-1-Formyl-pentyl)-carbamic acid (S)-2-cyclohex...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of human recombinant cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148291(((S)-1-Formyl-pentyl)-carbamic acid (S)-2-cyclohex...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of 10 uM Cbz-Phe-Arg-AMC binding to human cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148291(((S)-1-Formyl-pentyl)-carbamic acid (S)-2-cyclohex...)
Affinity DataIC50:  2.70nMAssay Description:Inhibitory concentration against human cathepsin K using 10 uM Cbz-Phe-Arg-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed