Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Corticotropin-releasing factor receptor 1' and Ligand = 'BDBM50293967'
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293967((R)-5-Chloro-3-(4-methoxy-2,5-dimethylphenylamino)...)
Affinity DataIC50:  0.880nMAssay Description:Displacement of [125I]-o-CRF from CRFR1 in rat frontal cortex after 2 hrs by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293967((R)-5-Chloro-3-(4-methoxy-2,5-dimethylphenylamino)...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]Tyr-ovine-CRF from CRF1 receptor in rat frontal cortex homogenate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed