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Found 2 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 1B1' and Ligand = 'BDBM50252405'
TargetCytochrome P450 1B1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50252405(CHEMBL556353 | Pifithrin-Alpha)
Affinity DataKi:  4.40nMAssay Description:Inhibition of recombinant CYP1B1 (unknown origin) expressed in supersomes coexpressing NADPH-CYP reductase using 7-ethoxyresorufin as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1B1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50252405(CHEMBL556353 | Pifithrin-Alpha)
Affinity DataIC50:  21nMAssay Description:Inhibition of CYP1B1 in TCDD-exposed human MCF-7 cells using ethoxyresorufin as substrate after 20 mins in presence of NADPH by spectrofluorimetric a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed