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Found 3 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 26A1' and Ligand = 'BDBM50342133'
TargetCytochrome P450 26A1(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50342133(Benzothiazol-2-yl-[4-((1S,2S)-2-dimethylamino-1-im...)
Affinity DataIC50:  10nMAssay Description:Inhibition of CYP26A1 in human MCF7 cell microsomes using [3H]ATRA after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 26A1(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50342133(Benzothiazol-2-yl-[4-((1S,2S)-2-dimethylamino-1-im...)
Affinity DataIC50:  10nMAssay Description:Inhibition of CYP26 in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 26A1(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50342133(Benzothiazol-2-yl-[4-((1S,2S)-2-dimethylamino-1-im...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human CYP26A1 assessed using [11,12-3H]ATRA as substrate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed