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Found 2 Enz. Inhib. hit(s) with Target = 'D(1B) dopamine receptor' and Ligand = 'BDBM50216047'
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216047(2-(4-(4-phenyl-1-piperazinyl)butyl)-1-isoindolinon...)
Affinity DataKi:  75.4nMAssay Description:Displacement of [3H]SCH 23390 from human Dopamine D5 receptor expressed in HEK293More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216047(2-(4-(4-phenyl-1-piperazinyl)butyl)-1-isoindolinon...)
Affinity DataKi:  137nMAssay Description:Antagonist activity at human Dopamine D5 receptor in HEK293 cells assessed as change in SKF 38393-induced intracellular calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed