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Found 3 Enz. Inhib. hit(s) with Target = 'DNA gyrase subunit A' and Ligand = 'BDBM50483022'
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
University Of Minnesota Medical School

Curated by ChEMBL
LigandPNGBDBM50483022(8-Methoxy Fluoroquinolone | CHEMBL1276635)
Affinity DataIC50:  120nMAssay Description:Inhibition of DNA supercoiling activity of Escherichia coli DNA gyrase gyrA A67S mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
University Of Minnesota Medical School

Curated by ChEMBL
LigandPNGBDBM50483022(8-Methoxy Fluoroquinolone | CHEMBL1276635)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of DNA supercoiling activity of Escherichia coli DNA gyrase gyrA G81C mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A(Escherichia coli (strain K12))
University Of Minnesota Medical School

Curated by ChEMBL
LigandPNGBDBM50483022(8-Methoxy Fluoroquinolone | CHEMBL1276635)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of DNA supercoiling activity of Escherichia coli DNA gyrase gyrA S83W mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed