Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM50253129'
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50253129(CHEMBL4066752)
Affinity DataKi:  0.154nMAssay Description:Positive allosteric modulation of human M4 receptor expressed in CHO cells co-expressing Gqi5 assessed as increase in acetylcholine-induced calcium m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50253129(CHEMBL4066752)
Affinity DataKi:  0.274nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50253129(CHEMBL4066752)
Affinity DataEC50:  0.540nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed