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Found 2 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase XIAP' and Ligand = 'BDBM50465645'
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50465645(CHEMBL4288478)
Affinity DataIC50:  37nMAssay Description:Displacement of AVPIAQKSEK-biotin from N-terminal His-tagged human recombinant XIAP BIR3 (253 to 347 residues) expressed in Escherichia coli BL21(DE3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
University Of California Riverside

Curated by ChEMBL
LigandPNGBDBM50465645(CHEMBL4288478)
Affinity DataKd:  86nMAssay Description:Binding affinity to N-terminal His-tagged human recombinant XIAP BIR3 (253 to 347 residues) expressed in Escherichia coli BL21(DE3) Gold by isotherma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed