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Found 6 Enz. Inhib. hit(s) with Target = 'Endoplasmin' and Ligand = 'BDBM21220'
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  110nMAssay Description:Inhibition of Grp94 (unknown origin)More data for this Ligand-Target Pair
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  110nMAssay Description:Displacement of FITC-geldanamycin from GRP94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetEndoplasmin(Canis familiaris)
Shandong University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKd:  2.80E+3nMAssay Description:Inhibition of N-terminal full length dog GRP94 (73 to 754 residues) expressed in Escherichia coli BL21(DE3) measured after 24 hrs by fluorescence pol...More data for this Ligand-Target Pair
TargetEndoplasmin(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKd:  200nMAssay Description:Displacement of [3H]NECA from GRP94 in porcine pancreas rough microsomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetEndoplasmin(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKd:  200nMAssay Description:Binding affinity to porcine pancreas rough microsomal GRP94 after 1 hrMore data for this Ligand-Target Pair
TargetEndoplasmin(Homo sapiens (Human))TBA
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKd:  530nMAssay Description:Displacement of FITC-geldanamycin from GRP94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair