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Found 3 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 1' and Ligand = 'BDBM50252049'
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252049((1S,3R)-1-aminopentane-1,3,5-tricarboxylic acid | ...)
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252049((1S,3R)-1-aminopentane-1,3,5-tricarboxylic acid | ...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human EAAT1 assessed as [3H]Asp uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50252049((1S,3R)-1-aminopentane-1,3,5-tricarboxylic acid | ...)
Affinity DataIC50:  3.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human EAAT1 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed