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Found 1 Enz. Inhib. hit(s) with Target = 'Gamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2' and Ligand = 'BDBM50166705'
LigandPNGBDBM50166705(2-(1-Benzenesulfonyl-cyclohexyl)-1,4-difluoro-benz...)
Affinity DataIC50:  98nMAssay Description:In vitro inhibition of gamma-secretase as amyloid peptide production in SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed