Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Gastrin/cholecystokinin type B receptor' and Ligand = 'BDBM50043548'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043548(1-(4-Chloro-phenyl)-3-{1-[2-(4-methyl-piperazin-1-...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of binding of [125I]-CCK-8 to the cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043548(1-(4-Chloro-phenyl)-3-{1-[2-(4-methyl-piperazin-1-...)
Affinity DataIC50:  2.60nMAssay Description:Ability to inhibit the binding of [125I]-gastrin to gastric glands in guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043548(1-(4-Chloro-phenyl)-3-{1-[2-(4-methyl-piperazin-1-...)
Affinity DataIC50:  8nMAssay Description:Ability to inhibit the binding of [125I]-CCK-8 to Cholecystokinin type B receptor in guinea pig cortex.More data for this Ligand-Target Pair
In DepthDetails Article