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Found 2 Enz. Inhib. hit(s) with Target = 'Ghrelin O-acyltransferase' and Ligand = 'BDBM289086'
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM289086(N-[(1 S)-2-[4-[2-[4-Amino-6-methyl-2-(trifluoromet...)
Affinity DataIC50:  69.5nMpH: 7.5Assay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO to obtain a ten-point dilution curve wi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM289086(N-[(1 S)-2-[4-[2-[4-Amino-6-methyl-2-(trifluoromet...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed