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Found 4 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Ligand = 'BDBM50316566'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50316566((+)-1-(2,3-dichlorophenyl)-2,2,2-trifluoro-1-(1-(4...)
Affinity DataIC50:  87nMAssay Description:Binding affinity to human glucocorticoid receptor by fluorescence polariztion competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50316566((+)-1-(2,3-dichlorophenyl)-2,2,2-trifluoro-1-(1-(4...)
Affinity DataIC50:  87nMAssay Description:Binding affinity to human glucocorticoid receptor by fluorescence polariztion competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50316566((+)-1-(2,3-dichlorophenyl)-2,2,2-trifluoro-1-(1-(4...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at glucocorticoid receptor in human fibroblast assessed as inhibition of IL-1-beta-induced IL6 production treated 1 hr before IL1-be...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50316566((+)-1-(2,3-dichlorophenyl)-2,2,2-trifluoro-1-(1-(4...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at glucocorticoid receptor in human MDA-kb2 cells transfected with MMTV-LUC assessed as induction of MMTV-LTR/promoter linked LUC ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed