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Found 5 Enz. Inhib. hit(s) with Target = 'Glycogen synthase kinase-3 beta' and Ligand = 'BDBM394123'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide GSM as substrate incubated for 30 mins in presence of ATP by Kinase-Glo ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  7.11E+3nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  7.11E+3nMAssay Description:Inhibition of human acrosin and control activity being 11.3 umol/min/mgMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  1.26E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Karolinska Institutet

Curated by ChEMBL
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  1.57E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent