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Found 3 Enz. Inhib. hit(s) with Target = 'Heparanase' and Ligand = 'BDBM50165612'
TargetHeparanase(Homo sapiens (Human))
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50165612((2-{4-[3-((E)-4-Bromo-phenyl)-acryloylamino]-pheny...)
Affinity DataIC50:  420nMAssay Description:Inhibition of recombinant HPSE (unknown origin) using fondaparinux as substrate incubated for 3 hrs in absence of light by WST1 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50165612((2-{4-[3-((E)-4-Bromo-phenyl)-acryloylamino]-pheny...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
"Sapienza" Universit£

Curated by ChEMBL
LigandPNGBDBM50165612((2-{4-[3-((E)-4-Bromo-phenyl)-acryloylamino]-pheny...)
Affinity DataIC50:  603nMAssay Description:Inhibition of heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed