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Found 2 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EHMT2' and Ligand = 'BDBM50300040'
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50300040(2-chloro-6,7-dimethoxy-N-(1-methylpiperidin-4-yl)q...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of G9a by Alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50300040(2-chloro-6,7-dimethoxy-N-(1-methylpiperidin-4-yl)q...)
Affinity DataIC50:  9.10E+6nMAssay Description:Inhibition of methyl transferase activity of G9a assessed as inhibition of H3K9 methylation by chemiluminescence based oxygen tunneling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed