Affinity DataKi: 800nMAssay Description:Displacement of [3H]-DPN from human KOR expressed in EE-HEK293 cell membranes by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Activity at human KOR expressed in EE-HEK293 cells assessed as pEC50 for effect on (-)U50,488H-induced response (Rvb = 6.2 +/- 0.04 No_unit)More data for this Ligand-Target Pair