Affinity DataKi: 28nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Displacement of [3H]U69593 from KOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]U-69593 from Opioid receptor kappa 1More data for this Ligand-Target Pair