Affinity DataKi: 720nMAssay Description:Inhibition of kappa opioid receptor (unknown origin) expressed in CHO cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) assessed as reduction in beta arrestin recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 8.75E+3nMAssay Description:Partial agonist activity at kappa opioid receptor (unknown origin) expressed in CHO cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair