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Found 3 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50528970'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50528970(CHEMBL4522339)
Affinity DataKi:  720nMAssay Description:Inhibition of kappa opioid receptor (unknown origin) expressed in CHO cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50528970(CHEMBL4522339)
Affinity DataEC50:  110nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) assessed as reduction in beta arrestin recruitmentMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50528970(CHEMBL4522339)
Affinity DataEC50:  8.75E+3nMAssay Description:Partial agonist activity at kappa opioid receptor (unknown origin) expressed in CHO cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed