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Found 4 Enz. Inhib. hit(s) with Target = 'Leukotriene B4 receptor 1/2' and Ligand = 'BDBM50036749'
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50036749(1-{5-ethyl-2-hydroxy-4-[6-methyl-6-(2H-1,2,3,4-tet...)
Affinity DataKi:  78nMAssay Description:In vitro inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50036749(1-{5-ethyl-2-hydroxy-4-[6-methyl-6-(2H-1,2,3,4-tet...)
Affinity DataIC50:  85nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50036749(1-{5-ethyl-2-hydroxy-4-[6-methyl-6-(2H-1,2,3,4-tet...)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of LTB4-induced human neutrophil CD11b/CD18 integrin up-regulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50036749(1-{5-ethyl-2-hydroxy-4-[6-methyl-6-(2H-1,2,3,4-tet...)
Affinity DataIC50:  2.87E+3nMAssay Description:LTB4-induced up-regulation of CD11b/CD18 in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article