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Found 277 Enz. Inhib. hit(s) with Target = 'Leukotriene B4 receptor 1/2'
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50013889((5S,6Z,8E,10E,12R,14Z)-5,12-dihydroxyicosa-6,8,10,...)
Affinity DataKi:  0.120nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50052021(4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-N,N-diis...)
Affinity DataKi:  1nMAssay Description:Inhibition of leukotriene B4 (LTB4) binding to its receptor on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231624(CHEMBL129703)
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231626(CHEMBL128013)
Affinity DataKi:  4.40nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231625(CHEMBL128067)
Affinity DataKi:  6.20nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50036743(CHEMBL60617 | Sodium salt of 4-Ethyl-5-[6-methyl-6...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50036750(2-ethoxy-4-ethyl-5-[6-methyl-6-(2H-1,2,3,4-tetraaz...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50001610(7-[3-(4-Acetyl-3-methoxy-2-propyl-phenoxy)-propoxy...)
Affinity DataKi:  15nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231631(CHEMBL128675)
Affinity DataKi:  21nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231603(CHEMBL128859)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231607(CHEMBL127218)
Affinity DataKi:  37nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212629(CHEMBL61542)
Affinity DataKi:  39nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231606(CHEMBL128755)
Affinity DataKi:  55nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212625(CHEMBL61919)
Affinity DataKi:  59nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231627(CHEMBL128888)
Affinity DataKi:  70nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231630(CHEMBL127274)
Affinity DataKi:  72nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212626(LY-255283)
Affinity DataKi:  77nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231628(CHEMBL130297)
Affinity DataKi:  77nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50036749(1-{5-ethyl-2-hydroxy-4-[6-methyl-6-(2H-1,2,3,4-tet...)
Affinity DataKi:  78nMAssay Description:In vitro inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231629(CHEMBL340649)
Affinity DataKi:  86nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212632(CHEMBL303109)
Affinity DataKi:  90nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212627(CHEMBL61920)
Affinity DataKi:  130nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212628(CHEMBL59656)
Affinity DataKi:  140nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231604(CHEMBL340386)
Affinity DataKi:  196nMAssay Description:Inhibition of [3H]LTB4 receptor binding in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212631(CHEMBL61913)
Affinity DataKi:  244nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212633(CHEMBL61770)
Affinity DataKi:  256nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50212630(CHEMBL61063)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of specific binding of [3H]-LTB4 to LTB4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50029464(5-(2-Carboxy-ethyl)-6-[3-(5-ethyl-4'-fluoro-2-hydr...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of LTB4-induced up-regulation of human neutrophil CD11b/CD18 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50029460(3-{3-[3-(5-Ethyl-4'-fluoro-2-hydroxy-biphenyl-4-yl...)
Affinity DataIC50:  1.80nMAssay Description:Tested for inhibition of specific binding of [3H]-LTB4 to guinea pig lung membranes expressing LTB4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50013889((5S,6Z,8E,10E,12R,14Z)-5,12-dihydroxyicosa-6,8,10,...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of specific binding of [3H]LTB4 to LTB4 receptor in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215854(CHEMBL301829)
Affinity DataIC50:  2nMAssay Description:Ability to inhibit LTB4-induced chemotaxis of isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215854(CHEMBL301829)
Affinity DataIC50:  2nMAssay Description:Ability to inhibit LTB4-induced chemotaxis of isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215854(CHEMBL301829)
Affinity DataIC50:  2.40nMAssay Description:Ability to inhibit LTB4-induced chemotaxis of isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231624(CHEMBL129703)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231606(CHEMBL128755)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231626(CHEMBL128013)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231625(CHEMBL128067)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215738(CHEMBL52675)
Affinity DataIC50:  3nMAssay Description:Ability to inhibit LTB4 binding to LTB receptors on isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50037218(1-((3S,4R)-3-Biphenyl-4-ylmethyl-4-hydroxy-chroman...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of leukotriene B4 (LTB4) binding to guinea pig spleenMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50029477(5-(2-Carboxy-ethyl)-6-[3-(5-ethyl-2-hydroxy-biphen...)
Affinity DataIC50:  3.40nMAssay Description:Tested for inhibition of specific binding of [3H]-LTB4 to human neutrophil expressing LTB4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50037218(1-((3S,4R)-3-Biphenyl-4-ylmethyl-4-hydroxy-chroman...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of LTB4 receptor induced chemotaxis of isolated human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50037218(1-((3S,4R)-3-Biphenyl-4-ylmethyl-4-hydroxy-chroman...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of LTB4 receptor induced chemotaxis of isolated human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50037218(1-((3S,4R)-3-Biphenyl-4-ylmethyl-4-hydroxy-chroman...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of LTB4 receptor induced chemotaxis of isolated human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231607(CHEMBL127218)
Affinity DataIC50:  4nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231631(CHEMBL128675)
Affinity DataIC50:  4nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215740(CHEMBL48906)
Affinity DataIC50:  4nMAssay Description:Ability to inhibit LTB4 binding to LTB receptors on isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215740(CHEMBL48906)
Affinity DataIC50:  4nMAssay Description:Ability to inhibit LTB4 binding to LTB receptors on isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50231603(CHEMBL128859)
Affinity DataIC50:  5nMAssay Description:Inhibition of [3H]LTB4 receptor binding in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215855(CHEMBL51467)
Affinity DataIC50:  5nMAssay Description:Ability to inhibit LTB4 binding to LTB receptors on isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1/2(Homo sapiens (Human))TBA
LigandPNGBDBM50215738(CHEMBL52675)
Affinity DataIC50:  5nMAssay Description:Ability to inhibit LTB4-induced chemotaxis of isolated human neutrophils.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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