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Found 4 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM135690'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135690(US10179804, Example 75 | US10632171, Peptide No. 7...)
Affinity DataKi:  0.600nMpH: 7.5Assay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135690(US10179804, Example 75 | US10632171, Peptide No. 7...)
Affinity DataKi:  0.600nMAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135690(US10179804, Example 75 | US10632171, Peptide No. 7...)
Affinity DataKi:  0.600nMAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135690(US10179804, Example 75 | US10632171, Peptide No. 7...)
Affinity DataKi:  0.600nM ΔG°:  -54.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent