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Found 3 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50168653'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50168653((R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(1-((2-...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of [125I]-AgRP(83¿132) (radioligand) binding to the hMC4R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50168653((R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(1-((2-...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50168653((R)-3-amino-N-(3-(2,4-dichlorophenyl)-1-(4-(1-((2-...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of [125I]NDP-MSH (radioligand) binding to the hMC4R stably expressed in HEK293 cells More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed