Affinity DataIC50: 70nMAssay Description:Inhibition of human MC4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]-NDP-R-MSH from human MC4R expressed in CHO cells after 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at human MC4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at human MC4R expressed in CHO cells assessed as cAMP releaseMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at human MC4R expressed in CHO cells assessed as increase of alpha-MSH-stimulated cAMP release pretreated for 10 mins before alpha-M...More data for this Ligand-Target Pair