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Found 4 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 14' and Ligand = 'BDBM50241114'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-Universit£T

Curated by ChEMBL
LigandPNGBDBM50241114(3-(2,4-Difluoro-phenylamino)-6H-dibenzo[b,e]oxepin...)
Affinity DataIC50:  239nMAssay Description:Inhibition of p38 alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-Universit£T

Curated by ChEMBL
LigandPNGBDBM50241114(3-(2,4-Difluoro-phenylamino)-6H-dibenzo[b,e]oxepin...)
Affinity DataIC50:  239nMAssay Description:Competitive inhibition of p38alpha MAP kinase (unknown origin) in presence of 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-Universit£T

Curated by ChEMBL
LigandPNGBDBM50241114(3-(2,4-Difluoro-phenylamino)-6H-dibenzo[b,e]oxepin...)
Affinity DataIC50:  240nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-Universit£T

Curated by ChEMBL
LigandPNGBDBM50241114(3-(2,4-Difluoro-phenylamino)-6H-dibenzo[b,e]oxepin...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of p38alpha MAP kinase in human whole blood assessed as inhibition of LPS-induced TNFalpha release by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed