Affinity DataKi: 11nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]DAMGO from MOR in guinea pig brain membranes measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
West Virginia University School Of Pharmacy
Curated by ChEMBL
West Virginia University School Of Pharmacy
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity was determined in a crude membrane preparation from guinea pig brain by displacement of [3H]DAMGO from Opioid receptor mu 1More data for this Ligand-Target Pair