Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50363079'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50363079(CHEMBL1944863 | N-(4-bromophenyl)-3,4,5-trimethoxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MRP1 expressed in MDCK cells assessed as calcein AM accumulation after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50363079(CHEMBL1944863 | N-(4-bromophenyl)-3,4,5-trimethoxy...)
Affinity DataIC50: >1.00E+5nMAssay Description:MDCK-MDR1 or MDCK-MRP1 cells (50,000 cells per well) were seeded into black CulturePlate (96-well plate) with 100 μL medium and allowed to becom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed