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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50549926'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Pipeline Therapeutics

Curated by ChEMBL
LigandPNGBDBM50549926(CHEMBL4783670)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Pipeline Therapeutics

Curated by ChEMBL
LigandPNGBDBM50549926(CHEMBL4783670)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed