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Found 2 Enz. Inhib. hit(s) with Target = 'Nicotinamide phosphoribosyltransferase' and Ligand = 'BDBM572570'
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM572570(1-[4-(4-Chloro-benzenesulfonyl)-phenyl]-3-(1H-pyra...)
Affinity DataEC50: <100nMAssay Description:NAMPT reaction was performed in 50 mM HEPES, pH 7.5, containing 5 mM MgCl2, 0.1% Prionex, 0.005% Tween 20, and 1 mM TCEP at room temperature in Grein...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM572570(1-[4-(4-Chloro-benzenesulfonyl)-phenyl]-3-(1H-pyra...)
Affinity DataEC50:  23nMAssay Description:Activation of human NAMPTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed