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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-beta' and Ligand = 'BDBM50121988'
Target
Nuclear receptor ROR-beta
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 4.10E+3nM
Assay Description:
Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...
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