Found 5 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50509558' 
Affinity DataIC50: 3nMAssay Description:Allosteric inhibition of recombinant His6-tagged RORgammat LBD (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as inhibition of bio...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataIC50: 3.80nMAssay Description:Activity at biotinylated 6His-tagged human RORgamma LBD (259 to 518 residues) assessed as induction of biotinylated SRC1 peptide recruitment incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human GAL4-fused RORgammat LBD transfected in Escherichia coli BL21(DE3) cell measured after 16 hrs by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Activity at RORgamma in human PBMC assessed as induction of IL17A production after 4 days by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Allosteric inhibition of yeast GAL4 DNA domain-fused RORgammat LBD (97 to 518 residues) (unknown origin) expressed in HEK293T cells after 20 to 22 hr...More data for this Ligand-Target Pair
