Found 6 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 4 group A member 1' and Ligand = 'BDBM50378798' TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 1.51E+3nMAssay Description:Binding affinity to NuR77-LBD receptor expressed in human BGC823 cellsMore data for this Ligand-Target Pair
3D Structure (crystal)TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 0.115nMAssay Description:Agonist activity at nuclear orphan receptor Nur77 expressed in human BGC823 cells co-transfected with fused GAL4-LBD assessed as transactivation afte...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 0.115nMAssay Description:Compound was tested for inhibitory activity against Dihydrofolate Reductase of rat liverMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 740nMAssay Description:Binding affinity to Nur77 receptor expressed in human BGC823 cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 0.278nMAssay Description:Inhibitory activity against Dihydrofolate reductase of Escherichia coliMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 4 group A member 1(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 0.278nMAssay Description:Agonist activity at nuclear orphan receptor Nur77 expressed in human BGC823 cells co-transfected with fused GAL4-Nur77 assessed as transactivation af...More data for this Ligand-Target Pair
