Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Oxysterols receptor LXR-beta' and Ligand = 'BDBM50012122'
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50012122(CHEMBL3263695)
Affinity DataIC50:  450nMAssay Description:Displacement of [3H]T0901317 from LXRbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50012122(CHEMBL3263695)
Affinity DataEC50:  1.90E+3nMAssay Description:Inverse agonist activity at human GAL4-fused LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed