Affinity DataIC50: 450nMAssay Description:Displacement of [3H]T0901317 from LXRbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Inverse agonist activity at human GAL4-fused LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-induced transcriptional activity af...More data for this Ligand-Target Pair