Found 11 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50145722'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 21.0nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Displacement of PPARalpha/delta agonist from human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.54E+3nMAssay Description:In vitro inhibition of mouse Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Transactivation activity for mouse Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Transactivation of Homo sapiens (human) PPARalpha assessed as luciferase activity by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Transcriptional activation of reporter assay by human Peroxisome proliferator activated receptor alpha in CV-1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARalpha DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARalpha DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Universidad Nacional Aut£Noma De M£Xico
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Transactivation activity for human Peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair