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Found 6 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50360740'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  8nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  5nMAssay Description:Agonist activity at GAL4-tagged PPARalpha ligand-binding domain (unknown origin) expressed in HEK293T cells incubated for 16 to 19 hrs by beta-lactam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  5nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at rat PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at mouse PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Canis familiaris)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  190nMAssay Description:Agonist activity at dog PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed