Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM50079260'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  284nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  301nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  423nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  949nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50079260(CHEMBL3416764)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity against pSG5-Gal4-tagged human PPAR-beta/delta ligand binding domain expressed in COS1 cells assessed as inhibition of GW501516-i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed