Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM50134237'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50:  598nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 3 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50:  907nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50134237(CHEMBL3740369)
Affinity DataIC50:  4.22E+3nMAssay Description:Binding affinity to GST-PPAR-beta/delta LBP (unknown origin) after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed