Found 4 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM28802' TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Co.
Bristol-Myers Squibb Co.
Affinity DataIC50: >1.50E+4nM EC50: 4.51E+3nMpH: 8.0 T: 2°CAssay Description:For PPARgamma, the percentage inhibition was calculated relative to rosiglitazone, which was used as the active site-specific competitive binder. Flu...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Co.
Bristol-Myers Squibb Co.
Affinity DataIC50: >9.84E+4nMAssay Description:Binding affinity to human GST-tagged PPAR-gamma LBD expressed in Escherichia coli BL21 after 30 mins in presence of fluorescein ligand FLA-A by fluor...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Co.
Bristol-Myers Squibb Co.
Affinity DataEC50: 4.51E+3nMAssay Description:Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Co.
Bristol-Myers Squibb Co.
Affinity DataEC50: >1.61E+3nMAssay Description:Agonist activity at full length human PPAR-gamma transfected in human HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
