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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50228360'
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228360(CHEMBL254814 | methyl 9-[1-(acetyloxyethyl)]-2-chl...)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228360(CHEMBL254814 | methyl 9-[1-(acetyloxyethyl)]-2-chl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50228360(CHEMBL254814 | methyl 9-[1-(acetyloxyethyl)]-2-chl...)
Affinity DataEC50:  160nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed