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Found 2 Enz. Inhib. hit(s) with Target = 'Prostacyclin receptor' and Ligand = 'BDBM357269'
TargetProstacyclin receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM357269(2-(((1s,4s)-4-((5- (ethylthio)-4-(2-fluoro-3- meth...)
Affinity DataEC50:  7nMAssay Description:Principle of the assay: The HTRF® assay kit was purchased from Cisbio-US, Inc. (Bedford, Mass.; Catalog #62AM4PEC). The HTRF® assay supported by the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstacyclin receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM357269(2-(((1s,4s)-4-((5- (ethylthio)-4-(2-fluoro-3- meth...)
Affinity DataEC50:  7nMAssay Description:The HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volume...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent