Affinity DataKi: 50nMAssay Description:In vitro binding affinity (agonistic) towards human CRTH2 receptor expressed in CHO cells; range 15 to 25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cells; range 25 nM to 8 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 389nMAssay Description:Partial antagonist activity at CRTH2 in human eosinophils assessed as inhibition of PGD2-induced shape change by FACS analysisMore data for this Ligand-Target Pair