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Found 3 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP2 subtype' and Ligand = 'BDBM50506546'
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))TBA
LigandPNGBDBM50506546(Omidenepag | UR-7276)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to EP2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))TBA
LigandPNGBDBM50506546(Omidenepag | UR-7276)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]prostaglandin E2 from human EP2 receptor expressed in HEK293 cell membranes after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))TBA
LigandPNGBDBM50506546(Omidenepag | UR-7276)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at recombinant human EP2 receptor expressed in HEK293 cells assessed as induction of cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed