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Found 6 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP3 subtype' and Ligand = 'BDBM35861'
TargetProstaglandin E2 receptor EP3 subtype(Mus musculus (Mouse))
Ono Pharmaceutical

LigandPNGBDBM35861(phenylpropanoic acid analogue, 5)
Affinity DataKi:  12nM EC50:  22nMAssay Description:Competitive binding studies were conducted using radiolabeled ligands and membrane fractions prepared from Chinese hamster ovary (CHO) cells stably e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Mus musculus (Mouse))
Ono Pharmaceutical

LigandPNGBDBM35861(phenylpropanoic acid analogue, 5)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]PGE2 from mouse EP3 receptor expressed in CHO cells after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Mus musculus (Mouse))
Ono Pharmaceutical

LigandPNGBDBM35861(phenylpropanoic acid analogue, 5)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at mouse EP3alpha receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium level ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Mus musculus (Mouse))
Ono Pharmaceutical

LigandPNGBDBM35861(phenylpropanoic acid analogue, 5)
Affinity DataIC50:  580nMAssay Description:Antagonist activity at mouse EP3alpha receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium level ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Mus musculus (Mouse))
Ono Pharmaceutical

LigandPNGBDBM35861(phenylpropanoic acid analogue, 5)
Affinity DataIC50:  580nMAssay Description:Antagonist activity at mouse EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium level after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Mus musculus (Mouse))
Ono Pharmaceutical

LigandPNGBDBM35861(phenylpropanoic acid analogue, 5)
Affinity DataIC50:  3.60E+3nMAssay Description:Antagonist activity at mouse EP3alpha receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium level ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed