Found 3 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP3 subtype' and Ligand = 'BDBM50248168'
Affinity DataIC50: 11.8nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of normal bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 23.7nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of 10% human serumMore data for this Ligand-Target Pair
Affinity DataEC50: 26.1nMAssay Description:Antagonist activity at human EP3-2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair