Found 4 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP4 subtype' and Ligand = 'BDBM50142488'
Affinity DataKi: 16nMAssay Description:Binding affinity was determined against prostanoid EP4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity to rat EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 460nMAssay Description:Agonist activity against recombinant prostanoid EP4 receptor stably transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Activity at rat EP4 transfected in HEK293 cells by cAMP accumulationMore data for this Ligand-Target Pair